SCHEMBL1920592

SCHEMBL1920592

CCCCc1ccccc1CBr

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LIPG Q9Y5X9 1/20 0.47
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
TLR8 Q9NR97 2/20 0.41
TYR P14679 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
ALOX5 P09917 1/20 0.38
PTGS2 P35354 1/20 0.38
HTR1A P08908 1/20 0.37
CTRC Q99895 1/20 0.36
BID P55957 3/20 0.36
MCL1 Q07820 3/20 0.36
BCL2L1 Q07817 2/20 0.36
BAK1 Q16611 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4459351 0.93 LIPG (0.55) LIPGTLR8NR1H2NR1H3ALOX5
SCHEMBL9579594 0.91 LIPG (0.58) LIPGCYP3A4TYRNR1H2NR1H3
SCHEMBL17027770 0.91 LIPG (0.58) LIPGCYP3A4TYRNR1H2NR1H3
SCHEMBL11354772 0.91 LIPG (0.58) LIPGCYP3A4TYRNR1H2NR1H3
SCHEMBL17027739 0.91 LIPG (0.58) LIPGCYP3A4TYRNR1H2NR1H3
SCHEMBL17027755 0.91 LIPG (0.58) LIPGCYP3A4TYRNR1H2NR1H3
SCHEMBL17027766 0.91 LIPG (0.58) LIPGCYP3A4TYRNR1H2NR1H3
SCHEMBL29520482 0.88 LIPG (0.56) LIPGCYP3A4CYP2D6CYP2C9TLR8
SCHEMBL245188 0.88 LIPG (0.56) LIPGCYP3A4CYP2D6CYP2C9TLR8
SCHEMBL8072359 0.86 LIPG (0.47) LIPGCYP3A4CYP2D6CYP2C9TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3105205-A1 PYRAZOLONE COMPOUNDS AND USES THEREOF Inception 2, Inc. (US) 2016-12-21 EP disclosed
EP-3022234-A1 SUBSTITUTED METALLOCENE CATALYSTS ExxonMobil Chemical Patents Inc. (US) 2016-05-25 EP disclosed
EP-2935228-A1 TRIAZOLONE COMPOUNDS AND USES THEREOF Inception 2, Inc. (US) 2015-10-28 EP disclosed
WO-2015123133-A1 PYRAZOLONE COMPOUNDS AND USES THEREOF INCEPTION 2, INC. (US) 2015-08-20 WO disclosed
WO-2015009479-A1 SUBSTITUTED METALLOCENE CATALYSTS EXXONMOBIL CHEMICAL PATENTS INC. (US) 2015-01-22 WO disclosed
WO-2014099503-A1 TRIAZOLONE COMPOUNDS AND USES THEREOF INCEPTION 2, INC. (US) 2014-06-26 WO disclosed
CN-101712828-B Ink jet ink, ink jet recording method, and ink cartridge CANON KK 2012-08-22 CN disclosed
EP-2326651-A1 BUPRENORPHINE ANALOGS Purdue Pharma LP (US) 2011-06-01 EP disclosed
CN-101712828-A Ink jet ink, ink jet recording method, and ink cartridge CANON KK 2010-05-26 CN disclosed
US-7674825-B2 Dicarboxylic acid derivatives with pharmaceutical properties BAYER AKTIENGESELLSCHAFT (DE) 2010-03-09 US disclosed
EP-0751767-A4 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE INC (US) 1997-12-10 EP disclosed
US-5637736-A Process for preparing 1-bromoalkylbenzene derivatives and intermediates thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-06-10 US disclosed
WO-1997015575-A1 PROTEIN KINASE C MODULATORS. Y. PROCYON PHARMACEUTICALS, INC. (US) 1997-05-01 WO disclosed
EP-0751767-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1997-01-08 EP disclosed
EP-0645458-A1 Chemoenzymatic process for production of S fenpropimorph CAFFARO S.p.A. Società per l'Industria Chimica ed Elettrochimica (IT) 1995-03-29 EP disclosed
EP-0637580-A1 Process for preparing 1-bromoalkylbenzene derivatives and intermediates thereof SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1995-02-08 EP disclosed
EP-0361040-A2 Odorless multi-valent metal modified products of salicylic acid copolymers, production processes thereof, and use thereof as color-developing agents for pressure-sensitive copying paper sheets MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-04-04 EP disclosed
EP-0355544-A2 Substituted decalin amines, method for their preparation and their use in pesticides BAYER AG (DE) 1990-02-28 EP disclosed
US-4277421-A P-TERT-BUTYLBENZAL BROMIDE HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-07 US disclosed
US-4261925-A Surfactants THE DOW CHEMICAL COMPANY (US) 1981-04-14 US disclosed