SCHEMBL1920805

SCHEMBL1920805

O=C(O)CN1CC(=O)c2ccc(N3CCN(C(=O)OCC4c5ccccc5-c5ccccc54)CC3)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.40
TMEM97 Q5BJF2 16/20 0.40
SIGMAR1 Q99720 16/20 0.40
HRH1 P35367 5/20 0.40
HRH3 Q9Y5N1 5/20 0.40
HRH2 P25021 4/20 0.40
HTR1A P08908 3/20 0.40
ADRA2A P08913 3/20 0.40
ADRA2B P18089 3/20 0.40
HTR2C P28335 3/20 0.40
ADRA2C P18825 2/20 0.40
HTR1E P28566 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2B P41595 2/20 0.40
ADRB1 P08588 1/20 0.40
DRD1 P21728 1/20 0.40
HTR1B P28222 1/20 0.40
SLC6A4 P31645 1/20 0.40
CYP2D6 P10635 2/20 0.39
DRD2 P14416 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1919543 0.89 PDK2 (0.40) PDK2TMEM97SIGMAR1HRH1HRH3
SCHEMBL8365081 0.80 TMEM97 (0.41) PDK2TMEM97SIGMAR1HRH1HRH3
SCHEMBL31505489 0.79 KDM4E (0.46) CYP2D6
SCHEMBL30481198 0.79 KDM4E (0.46) CYP2D6
SCHEMBL31398326 0.79 KDM4E (0.46) CYP2D6
SCHEMBL119822 0.79 KDM4E (0.46) CYP2D6
Water SCHEMBL4955373 0.78 KDM4E (0.45) HRH1HTR1AHTR2ACYP2D6DRD4
SCHEMBL1920229 0.76 KMT2A (0.41) PDK2CYP2D6DRD2DRD4SSTR1
SCHEMBL28078038 0.76 KDM4E (0.44) CYP2D6
SCHEMBL1920866 0.76 KDM4E (0.46) PDK2CYP2D6DRD2DRD4SSTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326666-A1 NEUROPEPTIDE-2 RECEPTOR (Y-2R) AGONISTS AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2011-06-01 EP disclosed
WO-2010031707-A1 NEUROPEPTIDE-2 RECEPTOR (Y-2R) AGONISTS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2010-03-25 WO disclosed