SCHEMBL19209848

SCHEMBL19209848

CC(C)c1c2cc(-c3nc(Nc4ccc(CN5CCNCC5)cn4)ncc3F)cnc2nn1C

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 17/20 0.68
CCND1 P24385 12/20 0.68
CDK4 P11802 9/20 0.68
CDK1 P06493 2/20 0.61
CDK2 P24941 2/20 0.61
CCNT1 O60563 1/20 0.61
CYP2C9 P11712 1/20 0.61
CCNB1 P14635 1/20 0.61
CCNE1 P24864 1/20 0.61
CYP2C19 P33261 1/20 0.61
CDK9 P50750 1/20 0.61
CDK5 Q00535 1/20 0.61
KCNH2 Q12809 1/20 0.61
CDK5R1 Q15078 1/20 0.61
DYRK2 Q92630 3/20 0.57
CCNA2 P20248 2/20 0.54
CCND3 P30281 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19231687 0.93 CDK6 (0.64) CDK6CCND1CDK4CDK1CDK2
SCHEMBL19209858 0.92 CDK6 (0.73) CDK6CCND1CDK4CDK1CDK2
SCHEMBL19209843 0.92 CDK6 (0.81) CDK6CCND1CDK4CDK1CDK2
SCHEMBL19231782 0.91 CDK6 (0.65) CDK6CCND1CDK4CDK1CDK2
SCHEMBL19231768 0.91 CDK6 (0.61) CDK6CCND1CDK4CDK1CDK2
SCHEMBL29518566 0.90 CDK6 (0.84) CDK6CCND1CDK4CDK1CDK2
SCHEMBL21208377 0.90 CDK6 (0.84) CDK6CCND1CDK4CDK1CDK2
SCHEMBL19231688 0.89 CDK6 (0.67) CDK6CCND1CDK4CDK1CDK2
Hydrochloric Acid SCHEMBL21201388 0.89 CDK6 (0.83) CDK6CCND1CDK4CDK1CDK2
SCHEMBL21208382 0.89 CDK6 (0.68) CDK6CCND1CDK4CDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133701-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 WO claimed
CN-108602799-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2021-08-03 CN disclosed
WO-2017133701-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 WO disclosed