SCHEMBL19209858

SCHEMBL19209858

CC(C)c1c2cc(-c3nc(Nc4ccc(CN5CCN(C)CC5)cn4)ncc3F)cnc2nn1C

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 18/20 0.73
CDK4 P11802 9/20 0.73
CCND1 P24385 7/20 0.73
CCND3 P30281 7/20 0.56
CDK2 P24941 4/20 0.56
CCNE2 O96020 3/20 0.56
CDK1 P06493 5/20 0.55
CCNA2 P20248 2/20 0.55
CCNT1 O60563 2/20 0.53
CCNB1 P14635 2/20 0.53
CCNE1 P24864 2/20 0.53
CDK9 P50750 2/20 0.53
CDK5 Q00535 2/20 0.53
KCNH2 Q12809 2/20 0.53
CDK5R1 Q15078 2/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
DYRK2 Q92630 3/20 0.52
CIT O14578 1/20 0.52
GAK O14976 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19209843 0.94 CDK6 (0.81) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19231688 0.94 CDK6 (0.67) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19209848 0.92 CDK6 (0.68) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19231827 0.92 CDK6 (0.64) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19231690 0.92 CDK6 (0.66) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19231681 0.90 CDK6 (0.75) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19209860 0.90 CDK6 (0.63) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19209882 0.90 CDK6 (0.65) CDK6CDK4CCND1CCND3CDK2
SCHEMBL22313803 0.90 CDK6 (0.89) CDK6CDK4CCND1CCND3CDK2
SCHEMBL19231782 0.90 CDK6 (0.65) CDK6CDK4CCND1CCND3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133701-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 WO claimed
CN-108602799-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2021-08-03 CN disclosed
WO-2017133701-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 WO disclosed