SCHEMBL19211458

SCHEMBL19211458

Fc1ccc(-n2cc(COc3cccc(Br)n3)nn2)cc1C(F)F

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RXRA P19793 20/20 0.78
GRIN1 Q05586 20/20 0.78
GRIN2B Q13224 20/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19219260 0.88 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19211468 0.87 RXRA (0.79) RXRAGRIN1GRIN2B
SCHEMBL19219261 0.84 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL28604820 0.82 RXRA (0.77) RXRAGRIN1GRIN2B
SCHEMBL19211440 0.80 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19211546 0.80 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19219259 0.79 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19219263 0.78 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL19219262 0.78 RXRA (1.00) RXRAGRIN1GRIN2B
SCHEMBL30030508 0.77 RXRA (0.50) RXRAGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071488-B Substituted 1,2, 3-triazoles as NR 2B-selective NMDA modulators 詹森药业有限公司 2021-08-13 CN disclosed
EP-3414233-A1 SUBSTITUTED 1,2,3-TRIAZOLES AS NR2B-SELECTIVE NMDA MODULATORS Janssen Pharmaceutica NV (BE) 2018-12-19 EP disclosed
WO-2017139428-A1 SUBSTITUTED 1,2,3-TRIAZOLES AS NR2B-SELECTIVE NMDA MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2017-08-17 WO disclosed