SCHEMBL1921440

SCHEMBL1921440

N#Cc1ccc(-c2ccnc(C(=O)NCC(=O)O)c2)cc1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 15/20 0.70
EGLN3 Q9H6Z9 3/20 0.62
FLT1 P17948 2/20 0.62
USP30 Q70CQ3 1/20 0.46
MMP2 P08253 1/20 0.45
GRM5 P41594 1/20 0.44
VEGFA P15692 1/20 0.43
EGLN2 Q96KS0 1/20 0.42
FTO Q9C0B1 1/20 0.42
PREP P48147 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14319654 0.90 EGLN1 (0.57) EGLN1EGLN3FLT1USP30MMP2
SCHEMBL1921655 0.86 EGLN1 (0.65) EGLN1EGLN3FLT1USP30GRM5
SCHEMBL14310050 0.84 EGLN1 (0.51) EGLN1EGLN3FLT1USP30MMP2
SCHEMBL10992192 0.83 EGLN1 (0.56) EGLN1EGLN3USP30EGLN2FTO
SCHEMBL17787716 0.83 KDM4E (0.53) EGLN1EGLN3FLT1USP30GRM5
SCHEMBL1921935 0.82 EGLN1 (0.70) EGLN1EGLN3FLT1VEGFA
SCHEMBL31226250 0.82 EGLN1 (0.68) EGLN1EGLN3FLT1VEGFA
SCHEMBL1921938 0.82 EGLN1 (0.68) EGLN1EGLN3FLT1VEGFA
SCHEMBL27751605 0.80 EGLN1 (0.46) EGLN1EGLN3FLT1USP30MMP2
SCHEMBL12979255 0.79 EGLN1 (0.61) EGLN1EGLN3FLT1VEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12478615-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2025-11-25 US disclosed
US-20240358691-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE WARNER CHILCOTT COMPANY, LLC (PR) 2024-10-31 US disclosed
US-11883386-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2024-01-30 US disclosed
US-20230201178-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE KREOS CAPITAL VII (UK) LIMITED (GB) 2023-06-29 US disclosed
US-20230201178-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE KREOS CAPITAL VII (UK) LIMITED (GB) 2023-06-29 US disclosed
EP-4095127-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE Akebia Therapeutics Inc. (US) 2022-11-30 EP disclosed
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2022-08-30 US disclosed
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2022-08-30 US disclosed
EP-3357911-B1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS INC (US) 2022-05-11 EP disclosed
EP-3357911-B1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS INC (US) 2022-05-11 EP disclosed
US-20100331374-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US disclosed
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US disclosed
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US disclosed
US-20100331374-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
EP-2044005-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE The Procter and Gamble Company (US) 2009-04-08 EP disclosed
WO-2008002576-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE THE PROCTER & GAMBLE COMPANY (US) 2008-01-03 WO disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885
US-11883386-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885
US-20240358691-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, EGLN2 EGLN1 6/4885EGLN3 2/4885FLT1 90/4885
US-20100331374-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885
US-12478615-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885
US-20230201178-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885FLT1 55/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.