SCHEMBL1922047

SCHEMBL1922047

COC(=O)Nc1ccc(-c2nc([C@H](Cc3ccc4c(c3)C[CH]C4)NC(=O)OC(C)(C)C)[nH]c2Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
F11 P03951 18/20 0.54
KLKB1 P03952 3/20 0.45
AAK1 Q2M2I8 1/20 0.38
CYP17A1 P05093 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1922048 0.90 F11 (0.53) F11KLKB1AAK1CYP17A1
SCHEMBL1196623 0.89 F11 (0.52) F11KLKB1AAK1CYP17A1
SCHEMBL1196982 0.88 F11 (0.51) F11KLKB1AAK1
SCHEMBL1196979 0.88 F11 (0.51) F11KLKB1AAK1
SCHEMBL1197002 0.85 F11 (0.58) F11KLKB1CYP17A1
SCHEMBL1196625 0.85 F11 (0.69) F11KLKB1
SCHEMBL1197016 0.83 F11 (0.60) F11KLKB1
SCHEMBL1195900 0.83 F11 (0.62) F11KLKB1
SCHEMBL1195903 0.83 F11 (0.62) F11KLKB1
SCHEMBL1197013 0.83 F11 (0.60) F11KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981854-B1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-06-01 EP disclosed