SCHEMBL19230302

SCHEMBL19230302

C=C(Nc1cccc(-c2cc(NC)c(=O)n(C)c2)c1C)c1cc2ccccc2s1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 12/20 0.46
BRD4 O60885 7/20 0.42
EGFR P00533 1/20 0.38
BMX P51813 1/20 0.38
JAK3 P52333 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL105874 0.82 BTK (0.54) BTKEGFRBMXJAK3
SCHEMBL1322596 0.73 BTK (0.73) BTKBMX
SCHEMBL20578298 0.73 BTK (0.59) BTKEGFRBMXJAK3
SCHEMBL20578299 0.72 BTK (0.56) BTKEGFRBMXJAK3
SCHEMBL20578293 0.71 BTK (0.59) BTKEGFRBMXJAK3
SCHEMBL20578196 0.70 BTK (0.65) BTKEGFRBMXJAK3
SCHEMBL20578265 0.69 BTK (0.57) BTKEGFRBMXJAK3
SCHEMBL12956109 0.69 BTK (0.59) BTKEGFRBMXJAK3
SCHEMBL20716894 0.67 BTK (0.54) BTK
SCHEMBL13044230 0.67 BTK (0.59) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133341-A1 NOVEL IRREVERSIBLE BRUTON'S TYROSINE KINASE INHIBITOR 中国科学院合肥物质科学研究院 2017-08-10 WO disclosed