SCHEMBL19233161

SCHEMBL19233161

CC(C)[C@H](C)Nc1nccc(N2CCNCC2)n1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 12/20 0.67
HRH3 Q9Y5N1 3/20 0.55
OGA O60502 1/20 0.46
CYP1A2 P05177 1/20 0.45
HSD17B10 Q99714 1/20 0.45
IDH1 O75874 1/20 0.45
CDK1 P06493 1/20 0.43
CDK4 P11802 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNA2 P20248 1/20 0.43
CCND1 P24385 1/20 0.43
CDK2 P24941 1/20 0.43
CCNA1 P78396 1/20 0.43
PLD1 Q13393 1/20 0.43
PRKD1 Q15139 2/20 0.42
PRKD2 Q9BZL6 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29935697 0.90 HRH4 (0.72) HRH4HRH3OGACYP1A2HSD17B10
SCHEMBL859700 0.90 HRH4 (0.72) HRH4HRH3OGACYP1A2HSD17B10
SCHEMBL19233404 0.84 HRH4 (0.81) HRH4HRH3OGACYP1A2HSD17B10
SCHEMBL13619336 0.82 HRH4 (0.66) HRH4HRH3CYP1A2HSD17B10PLD1
Hydrochloric Acid SCHEMBL26599748 0.81 HRH4 (0.64) HRH4HRH3CYP1A2HSD17B10PLD1
Hydrochloric Acid SCHEMBL30619112 0.81 HRH4 (0.64) HRH4HRH3CYP1A2HSD17B10PLD1
SCHEMBL1588650 0.81 HRH4 (1.00) HRH4HRH3OGA
SCHEMBL2575260 0.78 HRH4 (0.71) HRH4HRH3OGA
SCHEMBL13574661 0.77 HRH4 (0.80) HRH4HRH3OGAIDH1
SCHEMBL30834235 0.76 HRH3 (0.59) HRH4HRH3CYP1A2HSD17B10PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732087-B2 Diamino-pyridine, pyrimidine, and pyridazine modulators of the histamine H4 receptor JANSSEN PHARMACEUTICA N.V. (BE) 2017-08-15 US disclosed