SCHEMBL19250155

SCHEMBL19250155

COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)c(C)cc1C

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 19/20 0.85
ABL1 P00519 3/20 0.78
ABL2 P42684 2/20 0.78
FYN P06241 2/20 0.78
WEE2 P0C1S8 2/20 0.78
WEE1 P30291 2/20 0.78
PKMYT1 Q99640 2/20 0.78
BCR P11274 2/20 0.78
STK25 O00506 1/20 0.78
CIT O14578 1/20 0.78
RIOK3 O14730 1/20 0.78
MAP2K7 O14733 1/20 0.78
CHEK1 O14757 1/20 0.78
CASK O14936 1/20 0.78
GAK O14976 1/20 0.78
EPHB6 O15197 1/20 0.78
MAP3K13 O43283 1/20 0.78
MAP3K7 O43318 1/20 0.78
RIPK2 O43353 1/20 0.78
NUAK1 O60285 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23746826 0.93 SRC (0.88) SRCABL1ABL2FYNWEE2
SCHEMBL17460858 0.93 SRC (0.88) SRCABL1ABL2FYNWEE2
SCHEMBL20226049 0.88 SRC (0.78) SRCABL1ABL2FYNWEE2
SCHEMBL17855980 0.88 SRC (0.88) SRCABL1ABL2FYNWEE2
Bosutinib SCHEMBL158390 0.87 SRC (1.00) SRCABL1ABL2FYNWEE2
Bosutinib SCHEMBL29350234 0.87 SRC (1.00) SRCABL1ABL2FYNWEE2
Bosutinib SCHEMBL29428159 0.87 SRC (1.00) SRCABL1ABL2FYNWEE2
Bosutinib SCHEMBL19207253 0.87 SRC (1.00) SRCABL1ABL2FYNWEE2
SCHEMBL17505353 0.87 SRC (0.77) SRCABL1ABL2FYNWEE2
Bosutinib SCHEMBL29389315 0.87 SRC (1.00) SRCABL1ABL2FYNWEE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017134679-A1 NOVEL CRYSTALLINE POLYMORPHS OF 4-[(2.4-DICHIORO-5-METHOXVPHENVL)ANIINOL- 6-METHOXV-7-13-(4-METHYL-L-PIPERAZINVL)PROPOXVL-3-QUINOLINECARBONITRILE AND PROCESS FOR PREPARATION THEREOF MSN LABORATORIES PRIVATE LIMITED (IN) 2017-08-10 WO disclosed