SCHEMBL19251008

SCHEMBL19251008

CCCCC(C)(CCC)c1cnc(N)nc1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.33
TLR8 Q9NR97 6/20 0.33
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
PKM P14618 1/20 0.31
ESR1 P03372 2/20 0.31
ESR2 Q92731 2/20 0.31
TLR7 Q9NYK1 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21431386 0.93 CNR2 (0.34) NUDT1TLR8TLR7
SCHEMBL20017163 0.93 NUDT1 (0.33) NUDT1TLR8PKMTLR7
SCHEMBL18935611 0.93 NUDT1 (0.37) NUDT1PIK3R1PIK3CAESR1ESR2
SCHEMBL19251098 0.91 CNR2 (0.35) NUDT1TLR8TLR7
SCHEMBL20243849 0.91 CNR2 (0.35) NUDT1TLR8TLR7
SCHEMBL23957925 0.91 NUDT1 (0.34) NUDT1TLR8PKMTLR7
SCHEMBL19251245 0.89 CNR2 (0.35) NUDT1TLR8TLR7
SCHEMBL22752353 0.89 CNR2 (0.35) NUDT1TLR8TLR7
SCHEMBL19245805 0.89 CNR2 (0.35) NUDT1TLR8TLR7
SCHEMBL19135671 0.85 NUDT1 (0.35) NUDT1PIK3R1PIK3CAESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9993554-B2 Use of P13K Inhibitors for the Treatment of Obesity, Steatosis and ageing CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2018-06-12 US disclosed
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed