SCHEMBL19251223

SCHEMBL19251223

CCCCC(C)(CC)Oc1cncnc1

nearest known ligand 0.30

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22752567 0.93 CNR1 (0.34)
SCHEMBL19387704 0.90 CNR1 (0.33) CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL22752306 0.88 CNR1 (0.35)
SCHEMBL19251639 0.88 CNR1 (0.35)
SCHEMBL22752214 0.86 CNR2 (0.35) CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL19251373 0.86 CNR2 (0.35) CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL19251171 0.86 CNR2 (0.35) CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL22752291 0.85 CYP19A1 (0.35) CYP19A1
SCHEMBL19251152 0.82 CYP2D6 (0.32) CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL19251153 0.81 MAPT (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed