SCHEMBL19251639

SCHEMBL19251639

CCCCCCC(C)(CCCC)Oc1cncnc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.35
CNR2 P34972 3/20 0.35
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
ACAT1 P24752 1/20 0.31
SOAT1 P35610 1/20 0.31
GGPS1 O95749 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22752306 1.00 CNR1 (0.35) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL19251171 0.98 CNR2 (0.35) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL22752214 0.98 CNR2 (0.35) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL19251373 0.98 CNR2 (0.35) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL19387704 0.98 CNR1 (0.33) CNR1CNR2
SCHEMBL22752567 0.92 CNR1 (0.34) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL19251223 0.88 CYP1A2 (0.30)
SCHEMBL19251646 0.85 CNR2 (0.35) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL19251172 0.82 CNR2 (0.32) CNR1CNR2KDM4ETP53CYP3A4
SCHEMBL19251152 0.81 CYP2D6 (0.32) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed