SCHEMBL19251390

SCHEMBL19251390

CC(Nc1ncnc2[nH]cnc12)C1=Nc2ccccc2SN1c1cccc(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 13/20 0.38
PIK3CD O00329 12/20 0.38
PIK3CB P42338 5/20 0.37
PIK3CG P48736 5/20 0.37
PIK3CA P42336 3/20 0.37
CNR1 P21554 3/20 0.33
CNR2 P34972 3/20 0.33
SOS1 Q07889 2/20 0.32
KRAS P01116 1/20 0.32
CDK2 P24941 1/20 0.32
MAPK1 P28482 1/20 0.32
MAPK8 P45983 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CSNK1D P48730 1/20 0.32
CDK7 P50613 1/20 0.32
CCNH P51946 1/20 0.32
MNAT1 P51948 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19251385 0.90 PIK3CD (0.39) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251396 0.88 PIK3CD (0.45) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251398 0.84 PIK3CD (0.48) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251404 0.83 PIK3CD (0.49) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251631 0.80 PIK3R1 (0.60) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251611 0.78 PIK3CD (0.44) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19252623 0.78 PIK3CD (0.44) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251401 0.77 PIK3CD (0.49) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19252621 0.77 PIK3R1 (0.49) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA
SCHEMBL19251629 0.77 PIK3R1 (0.49) PIK3R1PIK3CDPIK3CBPIK3CGPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133655-A1 BENZOTHIAZINE AND BENZOTHIADIAZINE COMPOUNDS AND PREPARATION AND USE 浙江大学 2017-08-10 WO disclosed