SCHEMBL19252589

SCHEMBL19252589

CCCC(C)(C)c1cnc(SC)nc1

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19252593 0.89 KDM4E (0.35) KDM4EALDH1A1MAPTHPGDNPSR1
SCHEMBL22752529 0.86 CNR2 (0.42)
SCHEMBL19251007 0.84 MAPT (0.32) KDM4EALDH1A1MAPTHPGDNPSR1
SCHEMBL18744472 0.78 CNR2 (0.33)
SCHEMBL22752543 0.76 KDM4E (0.31) KDM4EALDH1A1MAPTHPGDNPSR1
SCHEMBL20878357 0.76 ESR1 (0.32)
SCHEMBL19069003 0.76 CNR2 (0.31)
SCHEMBL18935596 0.76 NUDT1 (0.37) KDM4EALDH1A1
SCHEMBL22752534 0.75 KDM4E (0.34) KDM4EALDH1A1MAPTHPGDNPSR1
SCHEMBL9906409 0.74 MEN1 (0.33) KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed