SCHEMBL19254058

SCHEMBL19254058

COc1ccc(C(OC[C@@H]2CC[C@H](n3cnc4c(=O)[nH]c(NC(=O)C(C)(C)CC(C)C(N)=O)nc43)O2)(c2ccccc2)c2ccc(OC)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMP P19971 9/20 0.43
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
HPGD P15428 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
ALB P02768 1/20 0.33
MAPK1 P28482 1/20 0.33
NT5E P21589 1/20 0.32
PDE9A O76083 2/20 0.32
HINT1 P49773 1/20 0.32
PDE2A O00408 1/20 0.31
PDE5A O76074 1/20 0.31
PDE4A P27815 1/20 0.31
PDE1B Q01064 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19505749 0.90 TYMP (0.48) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL13493900 0.88 TYMP (0.48) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL21473339 0.88 TYMP (0.48) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL19505895 0.87 TYMP (0.49) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL15488821 0.82 TYMP (0.45) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL15489089 0.81 TYMP (0.53) TYMPCYP1A2HPGDTAAR1ALDH1A1
SCHEMBL1697170 0.81 TYMP (0.43) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL15488822 0.80 TYMP (0.43) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL16451656 0.80 TYMP (0.43) TYMPKDM4ECYP1A2TAS1R3TAS1R1
SCHEMBL16451657 0.80 TYMP (0.43) TYMPKDM4ECYP1A2TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732112-B2 Synthesis of 2′,3′-dideoxynucleosides for automated DNA synthesis and pyrophosphorolysis activated polymerization Life Technologies Corporation (US) 2017-08-15 US disclosed