SCHEMBL19254478

SCHEMBL19254478

COc1cc(N(C)CCN(C)C)c(N)cc1Nc1nccc(Nc2cc(OC)c(OC)cc2C(C)=N)n1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.49
ALK Q9UM73 3/20 0.49
EML4 Q9HC35 2/20 0.48
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19254475 0.86 EGFR (0.49) EGFRALKEML4KCNH2
SCHEMBL19254476 0.84 EGFR (0.71) EGFRALKEML4KCNH2
SCHEMBL18386914 0.79 EGFR (0.47) EGFRALKKCNH2
SCHEMBL24445350 0.79 MAPK10 (0.48) EGFRALKEML4KCNH2
SCHEMBL22520183 0.79 EGFR (0.73) EGFRALKEML4
SCHEMBL19089365 0.78 EGFR (0.49) EGFRALKEML4
SCHEMBL29943919 0.78 EGFR (0.47) EGFRALKEML4KCNH2
SCHEMBL26101163 0.78 EGFR (0.47) EGFRALKEML4KCNH2
SCHEMBL21232425 0.77 EGFR (0.53) EGFRALKEML4
SCHEMBL24251743 0.76 EGFR (0.45) EGFRALKEML4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3205650-A1 EGFR INHIBITOR, AND PREPARATION AND APPLICATION THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2017-08-16 EP disclosed