SCHEMBL19256696

SCHEMBL19256696

COC(=O)c1nn(COC(=O)c2nn(C)cc2Br)cc1Br

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.48
RAB9A P51151 4/20 0.48
KDM4E B2RXH2 3/20 0.48
TP53 P04637 2/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
ALDH1A1 P00352 4/20 0.44
PKM P14618 2/20 0.44
SMN1; SMN2 Q16637 6/20 0.43
GAA P10253 1/20 0.41
LMNA P02545 4/20 0.41
ALPL P05186 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9948309 0.88 SMN1; SMN2 (0.51) NPC1RAB9AKDM4ETP53HSD17B10
SCHEMBL17375095 0.80 NPC1 (0.64) NPC1RAB9AKDM4ETP53HSD17B10
SCHEMBL858867 0.80 NPC1 (0.67) NPC1RAB9AKDM4EHSD17B10MEN1
SCHEMBL23850102 0.79 NPC1 (0.50) NPC1RAB9AKDM4ETP53HSD17B10
SCHEMBL31573749 0.75 NPC1 (0.46) NPC1RAB9AKDM4EHSD17B10MEN1
SCHEMBL31429362 0.75 NPC1 (0.46) NPC1RAB9AKDM4EHSD17B10MEN1
SCHEMBL16445216 0.75 ALDH1A1 (0.43) NPC1RAB9AKDM4EHSD17B10MEN1
SCHEMBL24211038 0.74 ALDH1A1 (0.47) NPC1RAB9AKDM4ETP53HSD17B10
SCHEMBL19879840 0.74 ALDH1A1 (0.42) NPC1RAB9AKDM4ETP53HSD17B10
SCHEMBL4443917 0.73 CNR2 (0.47) NPC1RAB9AKDM4ETP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3414241-B1 HALO-SUBSTITUTED PIPERIDINES AS OREXIN RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2022-05-04 EP disclosed
WO-2017139603-A1 HALO-SUBSTITUTED PIPERIDINES AS OREXIN RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2017-08-17 WO disclosed