SCHEMBL19256854

SCHEMBL19256854

C=CC(=O)N1CCC[C@@H](n2nc(-c3cc(C(=O)Nc4ccccc4)cs3)c3c(N)ncnc32)C1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 15/20 0.68
EGFR P00533 6/20 0.68
BTK Q06187 7/20 0.66
KCNH2 Q12809 3/20 0.66
JAK3 P52333 2/20 0.62
TEC P42680 3/20 0.62
BMX P51813 3/20 0.62
TXK P42681 2/20 0.62
LYN P07948 2/20 0.62
FGFR2 P21802 2/20 0.62
RIPK2 O43353 1/20 0.62
NR1I2 O75469 1/20 0.62
SLC22A3 O75751 1/20 0.62
LATS1 O95835 1/20 0.62
NUDT14 O95848 1/20 0.62
ABL1 P00519 1/20 0.62
ERBB2 P04626 1/20 0.62
LCK P06239 1/20 0.62
FYN P06241 1/20 0.62
PGR P06401 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28517769 0.94 ITK (0.65) ITKEGFRBTKKCNH2
SCHEMBL28517767 0.94 ITK (0.65) ITKEGFRBTKKCNH2
SCHEMBL28530486 0.93 ITK (0.62) ITKEGFRBTKKCNH2
SCHEMBL19257308 0.93 ITK (0.62) ITKEGFRBTKKCNH2
SCHEMBL28519894 0.91 ITK (0.64) ITKEGFRBTKKCNH2JAK3
SCHEMBL19257307 0.91 ITK (0.64) ITKEGFRBTKKCNH2JAK3
SCHEMBL19257305 0.87 EGFR (0.72) ITKEGFRBTKKCNH2JAK3
SCHEMBL19256932 0.87 EGFR (0.69) ITKEGFRBTKKCNH2JAK3
SCHEMBL19257235 0.87 EGFR (0.79) ITKEGFRBTKKCNH2JAK3
SCHEMBL28519532 0.87 EGFR (0.79) ITKEGFRBTKKCNH2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133630-A1 INHIBITOR OF BRUTON'S TYROSINE KINASE 北京盛诺基医药科技有限公司 2017-08-10 WO disclosed