SCHEMBL28530486

SCHEMBL28530486

C=CC(=O)N1CCCC(n2nc(-c3cc(C(=O)Nc4cccnc4)cs3)c3c(N)ncnc32)C1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITK Q08881 17/20 0.62
BTK Q06187 3/20 0.61
KCNH2 Q12809 2/20 0.60
EGFR P00533 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19257308 1.00 ITK (0.62) ITKBTKKCNH2EGFR
SCHEMBL19256854 0.93 ITK (0.68) ITKBTKKCNH2EGFR
SCHEMBL28517769 0.92 ITK (0.65) ITKBTKKCNH2EGFR
SCHEMBL28517767 0.92 ITK (0.65) ITKBTKKCNH2EGFR
SCHEMBL19256928 0.88 ITK (0.63) ITKBTKKCNH2EGFR
SCHEMBL28528837 0.88 ITK (0.63) ITKBTKKCNH2EGFR
SCHEMBL19257307 0.88 ITK (0.64) ITKBTKKCNH2EGFR
SCHEMBL28519894 0.88 ITK (0.64) ITKBTKKCNH2EGFR
SCHEMBL19257300 0.88 ITK (0.61) ITKBTKKCNH2EGFR
SCHEMBL28520057 0.88 ITK (0.61) ITKBTKKCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602834-B Bruton's tyrosine kinase inhibitor 北京盛诺基医药科技股份有限公司 2021-01-08 CN disclosed