SCHEMBL19258041

SCHEMBL19258041

C1=Cc2c(c3ccccc3n2-c2ccc(-c3cc(-c4ccccc4)cc(-c4ccccn4)n3)cc2)CN1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 12/20 0.34
DHODH Q02127 1/20 0.33
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CTSD P07339 1/20 0.32
CYP2C9 P11712 2/20 0.31
CYP1A2 P05177 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C19 P33261 1/20 0.31
PPP1CA P62136 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CCR1 P32246 1/20 0.31
CCR5 P51681 1/20 0.31
CCR8 P51685 1/20 0.31
ADORA3 P0DMS8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13569556 1.00 METAP1 (0.34) METAP1DHODHTSHRMAPK1HSD17B10
SCHEMBL19258569 0.97 METAP1 (0.35) METAP1DHODHCTSDCYP2C9CCR1
SCHEMBL13569543 0.95 METAP1 (0.32) METAP1DHODHCTSD
SCHEMBL13569500 0.92 MCL1 (0.33) METAP1TSHRHSD17B10CYP2C9CYP1A2
SCHEMBL13569600 0.91 METAP1 (0.34) METAP1CCR1CCR5CCR8
SCHEMBL13569478 0.90
SCHEMBL13569524 0.90 ADORA3 (0.30) ADORA3
SCHEMBL13569531 0.90 CCR1 (0.32) METAP1CCR1CCR5CCR8ADORA3
SCHEMBL13569630 0.89 ADORA3 (0.31) METAP1ADORA3
SCHEMBL13569467 0.89 HTR2C (0.35) METAP1MAPK1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2128159-B1 COMPOUND WHEREIN SUBSTITUTED BIPYRIDYL GROUP IS CONNECTED WITH PYRIDOINDOLE RING STRUCTURE THROUGH PHENYLENE GROUP, AND ORGANIC ELECTROLUMINESCENT DEVICE HODOGAYA CHEMICAL CO LTD (JP) 2017-08-16 EP disclosed