SCHEMBL19260285

SCHEMBL19260285

O=C1CCc2cc(Cl)c(F)cc2N1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 12/20 0.56
CA9 Q16790 1/20 0.46
KIF11 P52732 5/20 0.45
NPC1 O15118 1/20 0.43
MAPK13 O15264 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
PKLR P30613 1/20 0.41
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30888599 0.93 PKM (0.53) PKMCA9KIF11NPC1MAPK13
SCHEMBL4779437 0.93 PKM (0.53) PKMCA9KIF11NPC1MAPK13
SCHEMBL4104017 0.85 CA9 (0.52) PKMCA9KIF11NPC1MAPK13
SCHEMBL19278654 0.85 CA9 (0.52) PKMCA9KIF11NPC1MAPK13
SCHEMBL14780283 0.79 CA9 (0.46) PKMCA9KIF11NPC1MAPK13
SCHEMBL12992058 0.79 CA9 (0.54) PKMCA9KIF11NPC1MAPK13
SCHEMBL12559817 0.79 PKM (0.56) PKMCA9NPC1MAPK13MAPK12
SCHEMBL4104826 0.79 PKM (0.56) PKMCA9KIF11NPC1MAPK13
SCHEMBL21646067 0.79 CA9 (0.54) PKMCA9KIF11NPC1MAPK13
SCHEMBL18513614 0.79 PKM (0.47) PKMCA9KIF11NPC1MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3416633-B1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS UNIV ILLINOIS (US) 2025-07-23 EP disclosed
US-10456394-B2 Tetrahydroquinoline substituted hydroxamic acids as selective histone deacetylase 6 inhibitors THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2019-10-29 US disclosed
US-10456394-B2 Tetrahydroquinoline substituted hydroxamic acids as selective histone deacetylase 6 inhibitors THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2019-10-29 US disclosed
US-20190255046-A1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOS (US) 2019-08-22 US disclosed
US-20190255046-A1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOS (US) 2019-08-22 US disclosed
EP-3416633-A1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS The Board of Trustees of the University of Illinois (US) 2018-12-26 EP disclosed
WO-2017142883-A1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2017-08-24 WO disclosed
WO-2017142883-A1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2017-08-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190255046-A1 TETRAHYDROQUINOLINE SUBSTITUTED HYDROXAMIC ACIDS AS SELECTIVE HISTONE DEACETYLASE 6 INHIBITORS HDAC1, HDAC5, HDAC7 PKM 3014/4885CA9 2142/4885KIF11 2305/4885
US-10456394-B2 Tetrahydroquinoline substituted hydroxamic acids as selective histone deacetylase 6 inhibitors HDAC1, HDAC5, HDAC7 PKM 3014/4885CA9 2142/4885KIF11 2305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.