Formic Acid

Formic Acid

SCHEMBL19260728

COc1cc2cc3c(nc2cc1OCCCN1CCCC1)CCCC3.O=CO

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EHMT2 Q96KQ7 13/20 0.62
EHMT1 Q9H9B1 8/20 0.58
SPIN1 Q9Y657 3/20 0.48
TLR7 Q9NYK1 2/20 0.47
TLR9 Q9NR96 1/20 0.47
DNMT1 P26358 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29566009 0.94 EHMT2 (0.69) EHMT2EHMT1SPIN1TLR7TLR9
SCHEMBL19260596 0.94 EHMT2 (0.69) EHMT2EHMT1SPIN1TLR7TLR9
SCHEMBL19260582 0.92 EHMT2 (0.69) EHMT2EHMT1SPIN1TLR7TLR9
Formic Acid SCHEMBL19260670 0.79 ACHE (0.58) EHMT2EHMT1SPIN1TLR7TLR9
SCHEMBL20720679 0.78 EHMT2 (0.54) EHMT2EHMT1SPIN1TLR7TLR9
Formic Acid SCHEMBL19260744 0.78 EHMT2 (0.68) EHMT2SPIN1
Formic Acid SCHEMBL19260730 0.77 EHMT2 (0.55) EHMT2EHMT1TLR7TLR9DNMT1
Formic Acid SCHEMBL20720689 0.76 EHMT2 (0.69) EHMT2SPIN1DNMT1
Formic Acid SCHEMBL19260769 0.76 EHMT2 (0.57) EHMT2EHMT1SPIN1
SCHEMBL19260659 0.76 SPIN1 (0.57) EHMT2EHMT1SPIN1TLR7TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11254651-B2 Histone methyltransferase inhibitors GLOBAL BLOOD THERAPEUTICS, INC. (US) 2022-02-22 US disclosed
EP-3416963-B1 HISTONE METHYLTRANSFERASE INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2021-07-28 EP disclosed
US-20190047981-A1 HISTONE METHYLTRANSFERASE INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. 2019-02-14 US disclosed
EP-3416963-A1 HISTONE METHYLTRANSFERASE INHIBITORS Global Blood Therapeutics, Inc. (US) 2018-12-26 EP disclosed
WO-2017142947-A1 HISTONE METHYLTRANSFERASE INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. (US) 2017-08-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190047981-A1 HISTONE METHYLTRANSFERASE INHIBITORS EHMT1, EHMT2, BMI1 EHMT2 2/4885EHMT1 1/4885SPIN1 599/4885
US-11254651-B2 Histone methyltransferase inhibitors EHMT1, EHMT2, BMI1 EHMT2 2/4885EHMT1 1/4885SPIN1 599/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.