SCHEMBL19260858

SCHEMBL19260858

CC(C)OC(=O)C1=CN(C(=O)c2ccc(F)c(F)c2)CC(C)(C)c2c1[nH]c1cnccc21

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.80
ESR1 P03372 1/20 0.80
NR3C1 P04150 1/20 0.80
PGR P06401 1/20 0.80
NR3C2 P08235 1/20 0.80
AR P10275 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19260855 0.94 NR1H4 (0.80) NR1H4ESR1NR3C1PGRNR3C2
Turofexorate Isopropyl SCHEMBL274657 0.89 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2
Turofexorate Isopropyl SCHEMBL29823687 0.89 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2
Turofexorate Isopropyl SCHEMBL29382704 0.89 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL17883440 0.89 NR1H4 (0.80) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL17873357 0.87 NR1H4 (0.78) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL3738534 0.87 NR1H4 (0.83) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL3734487 0.86 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL4523649 0.85 NR1H4 (0.86) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL17873365 0.85 NR1H4 (0.74) NR1H4ESR1NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017143134-A1 FXR MODULATORS AND METHODS OF THEIR USE ALIOS BIOPHARMA, INC. (US) 2017-08-24 WO claimed
WO-2017143134-A1 FXR MODULATORS AND METHODS OF THEIR USE ALIOS BIOPHARMA, INC. (US) 2017-08-24 WO disclosed