SCHEMBL19267136

SCHEMBL19267136

CCNC(=O)c1c(O)n(-c2ccccn2)c(=O)n(Cc2ccccc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 2/20 0.45
PIK3CA P42336 1/20 0.43
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 4/20 0.42
LMNA P02545 3/20 0.42
TSHR P16473 2/20 0.42
PKM P14618 2/20 0.42
BRD4 O60885 1/20 0.42
TRPA1 O75762 1/20 0.42
EGLN1 Q9GZT9 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KCNH2 Q12809 1/20 0.41
ALOX12 P18054 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
USP2 O75604 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3420467 0.90 EGLN3 (0.56) EGLN3EGLN1
SCHEMBL3423631 0.83 MEN1 (0.50) ALDH1A1KDM4ELMNATSHRPKM
SCHEMBL19267278 0.81 EGLN3 (0.46) EGLN3ALDH1A1KDM4ELMNABRD4
SCHEMBL19267071 0.76 POLB (0.54) EGLN3ALDH1A1KDM4ELMNATSHR
SCHEMBL19267144 0.75 RGS4 (0.48) EGLN3LMNATSHRBRD4TP53
SCHEMBL3422070 0.73 EGLN3 (0.62) EGLN3EGLN1
SCHEMBL19267290 0.72 BRD4 (0.50) EGLN3PIK3CAALDH1A1KDM4ELMNA
SCHEMBL19267291 0.71 EGLN3 (0.43) EGLN3KDM4EBRD4EGLN1MEN1
SCHEMBL3421192 0.71 EGLN3 (0.69) EGLN3KDM4ELMNAEGLN1HTT
SCHEMBL18134558 0.71 EGLN3 (0.49) EGLN3KDM4ETRPA1EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037922-B9 PROLYL HYDROXYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2017-08-23 EP disclosed