SCHEMBL19286366

SCHEMBL19286366

N[C@@H](Cc1cccc(Cl)c1)C(O)N1CCN(C(=O)c2cc(F)ccc2F)CC1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.74
ALDH1A1 P00352 2/20 0.50
HTT P42858 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TSHR P16473 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
MDM2 Q00987 3/20 0.49
L3MBTL1 Q9Y468 2/20 0.47
SCN5A Q14524 1/20 0.45
SCN9A Q15858 1/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
PARP1 P09874 2/20 0.42
DPP4 P27487 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4909543 0.85 HDAC8 (1.00) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL17549802 0.85 HDAC8 (1.00) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL19887507 0.85 HDAC8 (1.00) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL4778030 0.79 HDAC8 (0.85) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL4905399 0.75 HDAC8 (0.80) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL4905417 0.75 HDAC8 (0.80) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL4795024 0.73 HDAC8 (0.76) HDAC8SMN1; SMN2MDM2KMT2AMEN1
SCHEMBL4905083 0.71 HDAC8 (0.62) HDAC8ALDH1A1HTTSMN1; SMN2KDM4E
SCHEMBL5013970 0.71 GPX4 (0.54) HDAC8
SCHEMBL4908436 0.71 HDAC8 (0.71) HDAC8ALDH1A1MDM2L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9745613-B2 Compounds, substrates and methods related to histone deacetylases THE BROAD INSTITUTE, INC. (US) 2017-08-29 US disclosed