SCHEMBL19292018

SCHEMBL19292018

Cn1ccc(-c2ccc(-c3cnc(CCCCCCC=O)[nH]3)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.40
KEAP1 Q14145 1/20 0.37
PDE10A Q9Y233 9/20 0.36
KMT2A Q03164 1/20 0.35
BRS3 P32247 1/20 0.35
SCN4A P35499 1/20 0.33
USP1 O94782 1/20 0.33
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19292474 0.89 CYP19A1 (0.38) CYP19A1KEAP1PDE10AKMT2ABRS3
SCHEMBL19292402 0.86 CYP19A1 (0.52) CYP19A1KEAP1PDE10AKMT2AMAPT
SCHEMBL15707115 0.83 PARP1 (0.40) CYP19A1KEAP1PDE10AKMT2ABRS3
SCHEMBL19292316 0.82 ACVR1 (0.37) PDE10A
SCHEMBL15707010 0.81 HDAC1 (0.42) CYP19A1BRS3
SCHEMBL19292264 0.80 CYP1A2 (0.43) CYP19A1PDE10ABRS3
SCHEMBL19292508 0.79 PDE10A (0.55) PDE10ABRS3
SCHEMBL19292260 0.79 PDE10A (0.42) PDE10AMAPT
SCHEMBL19292016 0.79 PDE10A (0.43) CYP19A1PDE10ABRS3
SCHEMBL19291980 0.79 PDE10A (0.37) PDE10ABRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2914589-B1 COMPOUNDS FOR USE IN THE TREATMENT OF PARASITIC DISEASES IRBM - SCIENCE PARK S P A (IT) 2017-08-30 EP disclosed