SCHEMBL19292016

SCHEMBL19292016

O=CCCCCCCc1ncc(-c2ccc(-c3ccccn3)cc2)[nH]1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 9/20 0.43
NPY5R Q15761 2/20 0.43
BRS3 P32247 3/20 0.42
NR1I2 O75469 1/20 0.42
NMBR P28336 1/20 0.42
GRPR P30550 1/20 0.42
KCNH2 Q12809 1/20 0.42
HPGDS O60760 1/20 0.39
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19292508 0.86 PDE10A (0.55) PDE10ABRS3HPGDS
SCHEMBL19292150 0.83 PDE10A (0.46) PDE10ANPY5RBRS3HPGDS
SCHEMBL19292513 0.82 BRS3 (0.45) PDE10ANPY5RBRS3NR1I2NMBR
SCHEMBL19291980 0.81 PDE10A (0.37) PDE10ABRS3
SCHEMBL19292309 0.81 HPGDS (0.45) PDE10ANPY5RBRS3HPGDSCYP2D6
SCHEMBL19292010 0.80 NLN (0.42) PDE10A
SCHEMBL19292018 0.79 CYP19A1 (0.40) PDE10ABRS3CYP19A1
SCHEMBL19292264 0.79 CYP1A2 (0.43) PDE10ABRS3CYP1A2CYP2D6CYP19A1
SCHEMBL19291976 0.79 PDE10A (0.43) PDE10ABRS3
SCHEMBL19292035 0.78 NPC1 (0.43) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2914589-B1 COMPOUNDS FOR USE IN THE TREATMENT OF PARASITIC DISEASES IRBM - SCIENCE PARK S P A (IT) 2017-08-30 EP disclosed