SCHEMBL19296286

SCHEMBL19296286

Cc1cc2cc(C(F)(F)F)ccc2cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
CYP2A6 P11509 1/20 0.52
CDK2 P24941 1/20 0.44
AKT1 P31749 1/20 0.44
BACE1 P56817 1/20 0.43
METAP2 P50579 1/20 0.43
THRB P10828 1/20 0.39
ABL1 P00519 1/20 0.38
PDE10A Q9Y233 1/20 0.37
GRM5 P41594 1/20 0.36
ESR1 P03372 1/20 0.36
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
SORT1 Q99523 3/20 0.36
KDM4E B2RXH2 1/20 0.36
NPBWR1 P48145 1/20 0.36
GAA P10253 1/20 0.35
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL803138 0.83 CYP1A2 (0.53) CYP1A2CYP2A6CDK2AKT1METAP2
SCHEMBL2749725 0.78 BACE1 (0.43) BACE1METAP2THRBESR1NOS3
SCHEMBL29964167 0.78 BACE1 (0.43) BACE1METAP2THRBESR1NOS3
SCHEMBL19877224 0.78 BACE1 (0.56) CDK2AKT1BACE1METAP2ABL1
SCHEMBL21083218 0.77 CYP1A2 (0.47) CYP1A2CYP2A6CDK2AKT1ESR1
SCHEMBL24796157 0.77 IDO1 (0.43) CYP1A2BACE1METAP2NPBWR1
SCHEMBL18899911 0.77 ABL1 (0.64) ABL1
SCHEMBL21920584 0.76 CYP1A2 (0.53) CYP1A2CYP2A6CDK2AKT1ABL1
SCHEMBL22002069 0.75 CYP1A2 (0.44) CYP1A2CYP2A6CDK2AKT1ESR1
SCHEMBL2320872 0.75 CYP1A2 (0.57) CYP1A2CYP2A6BACE1ABL1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170247393-A1 Aminoisoxazoline Compounds as Agonists of Alpha7-Nicotinic Acetylcholine Receptors FORUM PHARMACEUTICALS, INC. 2017-08-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170247393-A1 Aminoisoxazoline Compounds as Agonists of Alpha7-Nicotinic Acetylcholine Receptors CHRNA7, CHRNA5, CHRNA2 CYP1A2 943/4885CYP2A6 1601/4885CDK2 2825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.