SCHEMBL19308452

SCHEMBL19308452

CCCNC(=O)c1cc2ccccc2n1C

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.65
HDAC2 Q92769 1/20 0.65
MCL1 Q07820 1/20 0.58
HDAC3 O15379 1/20 0.57
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.52
HTR1A P08908 1/20 0.52
DRD2 P14416 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
DRD3 P35462 1/20 0.52
MAPT P10636 3/20 0.51
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HPGD P15428 1/20 0.51
GFER P55789 1/20 0.51
RXFP1 Q9HBX9 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16596183 0.89 HDAC1 (0.74) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL13753351 0.88 MCL1 (0.61) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL30174163 0.86 HDAC1 (0.66) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL3551679 0.86 HDAC1 (0.66) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL30174165 0.86 HDAC1 (0.66) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL24883665 0.86 HDAC1 (0.70) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL17373163 0.86 HDAC1 (0.62) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL14163703 0.85 HDAC1 (0.61) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL3554973 0.83 HDAC1 (0.60) HDAC1HDAC2MCL1HDAC3MEN1
SCHEMBL5669246 0.82 MCL1 (0.62) HDAC1HDAC2MCL1HDAC3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9751851-B2 Molecules and compositions that inhibit gram negative bacteria and their uses THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2017-09-05 US disclosed