SCHEMBL19320884

SCHEMBL19320884

COCc1ccccc1-c1sc2c(c1C(=O)O)CC(C)(C)CC2O

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.38
CACNA1H O95180 1/20 0.38
CACNA1I Q9P0X4 1/20 0.38
ESR1 P03372 1/20 0.34
PDK2 Q15119 1/20 0.32
P2RX3 P56373 3/20 0.32
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19325790 0.91 CACNA1G (0.30) CACNA1GCACNA1HCACNA1I
SCHEMBL19320881 0.81 CACNA1G (0.39) CACNA1GCACNA1HCACNA1IESR1P2RX3
SCHEMBL19140059 0.81 S1PR5 (0.33)
SCHEMBL19320874 0.80 PTPN1 (0.45) CACNA1GCACNA1HCACNA1IESR1PDK2
SCHEMBL19320826 0.80 CACNA1G (0.47) CACNA1GCACNA1HCACNA1IESR1CYP11B2
SCHEMBL19320875 0.78 CACNA1G (0.47) CACNA1GCACNA1HCACNA1IESR1CYP11B2
SCHEMBL19320882 0.74 ESR1 (0.33) CACNA1GCACNA1HCACNA1IESR1PDK2
SCHEMBL19320883 0.73 GSR (0.38) ESR1CYP11B2
SCHEMBL19320876 0.73 MAPT (0.44)
SCHEMBL19320828 0.73 CNR2 (0.39) CACNA1GCACNA1HCACNA1IESR1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170253607-A1 LONG-ACTING HIV PROTEASE INHIBITOR SHIONOGI & CO., LTD. (JP) 2017-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170253607-A1 LONG-ACTING HIV PROTEASE INHIBITOR CPN1, HAT1, PRSS1 CACNA1G 3034/4885CACNA1H 2888/4885CACNA1I 2662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.