SCHEMBL19331972

SCHEMBL19331972

COc1ccc(CNC2CCN(C(=O)OC(C)(C)C)CC2(C)C#N)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.48
STS P08842 2/20 0.47
MAPT P10636 1/20 0.45
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GPR119 Q8TDV5 1/20 0.40
BACE1 P56817 2/20 0.40
CTSD P07339 1/20 0.40
CTSE P14091 1/20 0.40
S1PR1 P21453 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MMP2 P08253 1/20 0.39
MMP13 P45452 1/20 0.39
NSD2 O96028 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19331914 0.91 EPHX2 (0.46) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL4732973 0.81 EPHX2 (0.61) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL16111394 0.81 EPHX2 (0.44) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL28611807 0.80 ALDH1A1 (0.54) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL27415157 0.80 ALDH1A1 (0.54) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL27415267 0.77 EPHX2 (0.46) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL21577641 0.77 EPHX2 (0.57) EPHX2STSMAPTALDH1A1MEN1
SCHEMBL18656011 0.76 EPHX2 (0.49) EPHX2STSMAPTALDH1A1TSHR
SCHEMBL19331898 0.75 TSHR (0.40) ALDH1A1TSHRMEN1KMT2AS1PR1
SCHEMBL27415228 0.75 TSHR (0.55) EPHX2STSMAPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017156177-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed
WO-2017156177-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed