SCHEMBL19331998

SCHEMBL19331998

COC(=O)CC1(NC(=O)C(F)(F)F)CCCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.38
PIK3R1 P27986 3/20 0.37
PIK3CA P42336 3/20 0.37
MMP2 P08253 1/20 0.35
MMP13 P45452 1/20 0.35
MMP14 P50281 1/20 0.35
ADAM17 P78536 1/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 3/20 0.34
CYP1A2 P05177 2/20 0.34
HPGD P15428 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
EPHX2 P34913 1/20 0.34
USP30 Q70CQ3 1/20 0.33
HDAC2 Q92769 1/20 0.33
EPHX1 P07099 1/20 0.33
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19331963 0.88 PIK3R1 (0.37) PIK3R1PIK3CAMMP2MMP13MMP14
SCHEMBL19331746 0.83 JAK2 (0.41) PIK3R1PIK3CAMMP2MMP13MMP14
SCHEMBL19331794 0.81 PIK3R1 (0.36) PIK3R1PIK3CAMMP2MMP13MMP14
SCHEMBL5568440 0.79 HDAC2 (0.37) PIK3R1PIK3CAEPHX2HDAC2USP2
SCHEMBL5567244 0.79 HDAC2 (0.39) PIK3R1PIK3CAEPHX2HDAC2USP2
SCHEMBL19331906 0.76 HPGD (0.38) CNR2PIK3R1PIK3CAMMP2MMP13
SCHEMBL1586974 0.73 EPHX2 (0.43) MMP13ADAM17MAPTEPHX2HDAC2
SCHEMBL429808 0.73 CNR2 (0.42) CNR2PIK3R1PIK3CAADAM17ALDH1A1
SCHEMBL1684623 0.72 EPHX2 (0.40) MMP13ADAM17MAPTEPHX2HDAC2
SCHEMBL25169698 0.71 USP2 (0.43) CNR2ALDH1A1HPGDEPHX2EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017156177-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed
WO-2017156177-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed