SCHEMBL19331963

SCHEMBL19331963

CNC(=O)CC1(NC(=O)C(F)(F)F)CCCN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3R1 P27986 3/20 0.37
PIK3CA P42336 3/20 0.37
ADAM17 P78536 2/20 0.35
MMP2 P08253 1/20 0.35
MMP13 P45452 1/20 0.35
MMP14 P50281 1/20 0.35
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.33
EPHX2 P34913 1/20 0.33
USP30 Q70CQ3 1/20 0.33
HDAC2 Q92769 1/20 0.32
EPHX1 P07099 1/20 0.32
USP2 O75604 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
CYP11B2 P19099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19331998 0.88 CNR2 (0.38) PIK3R1PIK3CAADAM17MMP2MMP13
SCHEMBL19331746 0.82 JAK2 (0.41) PIK3R1PIK3CAADAM17MMP2MMP13
SCHEMBL19331794 0.81 PIK3R1 (0.36) PIK3R1PIK3CAADAM17MMP2MMP13
SCHEMBL19331734 0.79 HPGD (0.37) PIK3R1PIK3CAADAM17MMP2MMP13
SCHEMBL5567244 0.78 HDAC2 (0.39) PIK3R1PIK3CAEPHX2HDAC2USP2
SCHEMBL5568440 0.78 HDAC2 (0.37) PIK3R1PIK3CAEPHX2HDAC2USP2
SCHEMBL1586974 0.72 EPHX2 (0.43) ADAM17MMP13MAPTEPHX2HDAC2
SCHEMBL24080972 0.72 USP2 (0.42) ADAM17MMP2MMP13MMP14HPGD
SCHEMBL1684623 0.72 EPHX2 (0.40) ADAM17MMP13MAPTEPHX2HDAC2
SCHEMBL19331967 0.71 HPGD (0.36) PIK3R1PIK3CAADAM17MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017156177-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed
WO-2017156177-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed