SCHEMBL19337026

SCHEMBL19337026

COc1cc(F)c([N+](=O)[O-])cc1Nc1nccc(C(=N)c2ccccc2NC(C)C)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.41
CDK9 P50750 1/20 0.41
RXFP1 Q9HBX9 1/20 0.39
MAPK8 P45983 5/20 0.39
GSK3B P49841 5/20 0.39
PTK2 Q05397 3/20 0.39
PLK1 P53350 2/20 0.39
GSK3A P49840 2/20 0.39
ALK Q9UM73 2/20 0.39
CDC7 O00311 1/20 0.39
PLK4 O00444 1/20 0.39
CHEK1 O14757 1/20 0.39
DCLK1 O15075 1/20 0.39
CHUK O15111 1/20 0.39
PDPK1 O15530 1/20 0.39
DAPK3 O43293 1/20 0.39
DYRK3 O43781 1/20 0.39
JAK2 O60674 1/20 0.39
ROCK2 O75116 1/20 0.39
PRKD3 O94806 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19336964 0.91 CCNT1 (0.43) CCNT1CDK9MAPK8GSK3BPTK2
SCHEMBL19337022 0.85 EGFR (0.47) ALKINSRKDRJAK3EGFR
SCHEMBL32681522 0.80 CCNT1 (0.42) CCNT1CDK9MAPK8GSK3BGSK3A
SCHEMBL22509271 0.79 PTK2 (0.48) CCNT1CDK9MAPK8GSK3BPTK2
SCHEMBL22994859 0.79 CCNT1 (0.39) CCNT1CDK9MAPK8GSK3BPTK2
SCHEMBL32681474 0.78 KMT2A (0.46) CCNT1CDK9MAPK8GSK3BGSK3A
SCHEMBL19336965 0.76 EGFR (0.48) ALKINSRKDRJAK3EGFR
SCHEMBL29597402 0.75 KMT2A (0.47) CCNT1CDK9MAPK1EGFRMEN1
SCHEMBL30948589 0.75 CCNT1 (0.42) CCNT1CDK9MAPK8GSK3BPTK2
SCHEMBL32681483 0.75 KMT2A (0.41) CCNT1CDK9GSK3BGSK3AEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3216786-A1 PYRIMIDINE OR PYRIDINE COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USES THEREOF Shanghai Shaletech Technology Co., Ltd. (CN) 2017-09-13 EP disclosed