SCHEMBL19337095

SCHEMBL19337095

C=CC(=O)Nc1cc(Nc2nccc(Nc3ccccc3N(C)[SH](=O)=O)n2)c(OC)cc1N(C)CCN(C)C

nearest known ligand 0.77

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.77
ALK Q9UM73 3/20 0.77
EML4 Q9HC35 2/20 0.76
KCNH2 Q12809 2/20 0.64
PTK2 Q05397 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23865682 0.89 EGFR (0.71) EGFRALKEML4KCNH2PTK2
SCHEMBL19089663 0.88 EGFR (0.82) EGFRALKEML4KCNH2
SCHEMBL19337136 0.88 EGFR (0.77) EGFRALKEML4KCNH2PTK2
SCHEMBL19337163 0.87 EGFR (0.76) EGFRALKEML4KCNH2PTK2
SCHEMBL27237904 0.87 EGFR (0.80) EGFRALKEML4KCNH2PTK2
SCHEMBL22497616 0.87 EGFR (1.00) EGFRALKEML4
SCHEMBL19337177 0.87 EGFR (0.76) EGFRALKEML4KCNH2
SCHEMBL30222929 0.87 EGFR (0.79) EGFRALKEML4KCNH2PTK2
SCHEMBL20655381 0.86 EGFR (0.73) EGFRALKEML4
SCHEMBL27237906 0.85 EGFR (0.77) EGFRALKEML4KCNH2PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3885344-A2 PYRIMIDINE COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USES THEREOF InventisBio Co., Ltd. (CN) 2021-09-29 EP disclosed
EP-3216786-A1 PYRIMIDINE OR PYRIDINE COMPOUNDS, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USES THEREOF Shanghai Shaletech Technology Co., Ltd. (CN) 2017-09-13 EP disclosed