SCHEMBL19337490

SCHEMBL19337490

COc1cc(C(=O)NC(=S)Nc2cccc(NC(=O)c3ccc4ccccc4c3)c2)cc(C)c1OC

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 12/20 0.70
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
NQO2 P16083 1/20 0.54
CASP3 P42574 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
ALDH1A1 P00352 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
ALOX12 P18054 1/20 0.54
CYP2C19 P33261 1/20 0.54
TDP1 Q9NUW8 2/20 0.52
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
POLB P06746 1/20 0.52
RECQL P46063 1/20 0.52
BLM P54132 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12129855 0.94 SMO (0.78) SMONPC1RAB9ANQO2CASP3
SCHEMBL12129883 0.84 SMO (0.78) SMONPC1RAB9ANQO2CASP3
SCHEMBL12129870 0.83 SMO (0.83) SMONPC1RAB9AALDH1A1CYP2C9
SCHEMBL1335388 0.83 RAB9A (0.70) SMONPC1RAB9ACASP3SENP7
SCHEMBL12129826 0.83 SMO (0.83) SMONPC1RAB9AALDH1A1CYP2C9
SCHEMBL29390703 0.82 SMO (1.00) SMONPC1RAB9AALDH1A1CYP2C9
SCHEMBL12129860 0.82 SMO (1.00) SMONPC1RAB9AALDH1A1CYP2C9
SCHEMBL8211832 0.82 SMO (0.62) SMONPC1RAB9ANQO2CASP3
SCHEMBL19337622 0.82 SMO (0.82) SMONPC1RAB9AALDH1A1CYP2C9
SCHEMBL12129833 0.82 SMO (0.82) SMONPC1RAB9ACASP3SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2291352-B1 N-ACYLTHIOUREA AND N-ACYLUREA INHIBITORS OF THE HEDGEHOG PROTEIN SIGNALLING PATHWAY CENTRE NAT RECH SCIENT (FR) 2017-09-13 EP disclosed