SCHEMBL1934409

SCHEMBL1934409

CC1N[C@H](C(=O)O)Cc2c1[nH]c1ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.74
TSHR P16473 2/20 0.74
HSD17B10 Q99714 2/20 0.74
HTT P42858 1/20 0.74
CYP2D6 P10635 3/20 0.71
MAPK1 P28482 1/20 0.71
MEN1 O00255 5/20 0.70
KMT2A Q03164 5/20 0.70
ALDH1A1 P00352 4/20 0.70
MAPT P10636 1/20 0.70
HPGD P15428 1/20 0.70
CYP2C19 P33261 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
ALOX12 P18054 1/20 0.60
ALOX15 P16050 1/20 0.57
CCKBR P32239 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28642718 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL28662843 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL29379056 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL31310810 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL5680135 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL504399 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL18207946 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL10843678 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL1934152 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6
SCHEMBL4762341 1.00 KDM4E (0.74) KDM4ETSHRHSD17B10HTTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108948001-A The synthetic route of 1R, 3S-1- methyl tetrahydro-beta-carboline -3- carboxylic acid, anti-thrombus activity and application 首都医科大学 2018-12-07 CN claimed
EP-2332539-A1 PHARMACEUTICAL PREPARATION, FOOD OR BEVERAGE HAVING INHIBITORY ACTIVITY ON SEROTONIN TRANSPORTER Suntory Holdings Limited (JP) 2011-06-15 EP claimed
CN-108948001-A The synthetic route of 1R, 3S-1- methyl tetrahydro-beta-carboline -3- carboxylic acid, anti-thrombus activity and application 首都医科大学 2018-12-07 CN disclosed
CN-107686482-A New heptacyclic compound, it is synthesized, activity rating and application 首都医科大学 2018-02-13 CN disclosed
WO-2004113336-A1 CARBOLINE AND BETACARBOLINE DERIVATIVES FOR USE AS HDAC ENZYME INHIBITORS CHROMA THERAPEUTICS LIMITED (GB) 2004-12-29 WO disclosed