SCHEMBL1935628

SCHEMBL1935628

COCCCNC(=O)c1cccs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 1.00
KDM4E B2RXH2 2/20 0.76
SMN1; SMN2 Q16637 3/20 0.74
HPGD P15428 4/20 0.67
NPC1 O15118 3/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2C9 P11712 2/20 0.62
CYP2C19 P33261 2/20 0.62
POLB P06746 1/20 0.62
ALOX15 P16050 1/20 0.62
LMNA P02545 2/20 0.61
HTT P42858 1/20 0.61
ALDH1A1 P00352 4/20 0.60
CYP3A4 P08684 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
RAB9A P51151 2/20 0.59
THRB P10828 1/20 0.58
TSHR P16473 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2330242 0.90 GAA (0.82) GAAKDM4ESMN1; SMN2HPGDNPC1
SCHEMBL6127192 0.85 KDM4E (0.89) GAAKDM4ESMN1; SMN2NPC1CYP1A2
SCHEMBL4045277 0.84 KDM4E (0.81) GAAKDM4ESMN1; SMN2NPC1CYP1A2
SCHEMBL5246151 0.83 KDM4E (0.78) GAAKDM4ESMN1; SMN2NPC1CYP1A2
SCHEMBL12491925 0.83 GAA (0.70) GAAKDM4ESMN1; SMN2HPGDNPC1
SCHEMBL18197872 0.83 KDM4E (0.84) GAAKDM4ESMN1; SMN2HPGDNPC1
SCHEMBL18906066 0.82 KDM4E (0.83) GAAKDM4ESMN1; SMN2NPC1CYP1A2
SCHEMBL3814103 0.82 GAA (0.69) GAAKDM4ESMN1; SMN2HPGDNPC1
SCHEMBL8966500 0.81 GAA (0.68) GAAKDM4ESMN1; SMN2HPGDNPC1
SCHEMBL6928579 0.81 KDM4E (0.76) GAAKDM4ESMN1; SMN2NPC1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509602-A1 PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS CK2 INHIBITORS Cylene Pharmaceuticals, Inc. (US) 2012-10-17 EP disclosed
WO-2011068667-A1 PYRAZOLOPYRIMIDINES AND RELATED HETEROCYCLES AS CK2 INHIBITORS CYLENE PHARMACEUTICALS, INC. (US) 2011-06-09 WO disclosed