SCHEMBL19357643

SCHEMBL19357643

N#Cc1cc(Cl)ccc1-c1cccc2c1CN(C#N)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TEAD1 P28347 5/20 0.39
TEAD4 Q15561 5/20 0.39
TEAD2 Q15562 5/20 0.39
TEAD3 Q99594 1/20 0.39
HSD17B3 P37058 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CNR1 P21554 3/20 0.34
CNR2 P34972 3/20 0.34
SCN9A Q15858 2/20 0.34
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSK P43235 1/20 0.33
CYP2A6 P11509 1/20 0.33
OTUD7B Q6GQQ9 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29710124 1.00 TEAD1 (0.39) TEAD1TEAD4TEAD2TEAD3HSD17B3
SCHEMBL19357743 0.86 TEAD1 (0.41) TEAD1TEAD4TEAD2TEAD3CTSL
SCHEMBL19357844 0.84 TEAD1 (0.42) TEAD1TEAD4TEAD2TEAD3SCN9A
SCHEMBL29710034 0.84 TEAD1 (0.42) TEAD1TEAD4TEAD2TEAD3SCN9A
SCHEMBL29710091 0.84 BTK (0.44) TEAD1TEAD4TEAD2TEAD3HSP90AA1
SCHEMBL19357751 0.84 BTK (0.44) TEAD1TEAD4TEAD2TEAD3HSP90AA1
SCHEMBL29710088 0.83 TEAD1 (0.47) TEAD1TEAD4TEAD2TEAD3CTSL
SCHEMBL19357728 0.83 TEAD1 (0.47) TEAD1TEAD4TEAD2TEAD3CTSL
SCHEMBL29710074 0.81 USP7 (0.46) TEAD1TEAD4TEAD2TEAD3SCN9A
SCHEMBL19358029 0.81 USP7 (0.46) TEAD1TEAD4TEAD2TEAD3SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108698992-B 2-cyanoisoindoline derivatives for the treatment of cancer 特殊治疗有限公司 2022-04-19 CN claimed
EP-3429994-B1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LTD (GB) 2021-06-16 EP claimed
US-10683269-B2 2-cyanoisoindoline derivatives for treating cancer MISSION THERAPEUTICS LIMITED (GB) 2020-06-16 US claimed
EP-3429994-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER Mission Therapeutics Limited (GB) 2019-01-23 EP claimed
US-20190010122-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2019-01-10 US claimed
WO-2017158388-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2017-09-21 WO claimed
CN-108698992-B 2-cyanoisoindoline derivatives for the treatment of cancer 特殊治疗有限公司 2022-04-19 CN disclosed
EP-3429994-B1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LTD (GB) 2021-06-16 EP disclosed
US-10683269-B2 2-cyanoisoindoline derivatives for treating cancer MISSION THERAPEUTICS LIMITED (GB) 2020-06-16 US disclosed
EP-3429994-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER Mission Therapeutics Limited (GB) 2019-01-23 EP disclosed
US-20190010122-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2019-01-10 US disclosed
WO-2017158388-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER MISSION THERAPEUTICS LIMITED (GB) 2017-09-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190010122-A1 2-CYANOISOINDOLINE DERIVATIVES FOR TREATING CANCER USP7, USP47, USP2 TEAD1 2150/4885TEAD4 2517/4885TEAD2 2851/4885
US-10683269-B2 2-cyanoisoindoline derivatives for treating cancer USP7, USP47, USP2 TEAD1 2150/4885TEAD4 2517/4885TEAD2 2851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.