SCHEMBL19360362

SCHEMBL19360362

COC(=O)c1ccc2[nH]c(Cc3ccccc3OC(F)(F)F)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.46
F2 P00734 2/20 0.46
FFAR1 O14842 1/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
GPR84 Q9NQS5 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
PPARG P37231 2/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
KIF11 P52732 1/20 0.39
KDR P35968 2/20 0.39
EPHX2 P34913 1/20 0.39
RORC P51449 1/20 0.38
PDE9A O76083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360304 0.88 F2 (0.47) F2GPR84KDM4EALDH1A1HTT
SCHEMBL19360428 0.85 F2 (0.47) F2FFAR1ROCK2ROCK1GPR84
SCHEMBL19360372 0.83 F2 (0.49) F2GPR84KDM4EALDH1A1L3MBTL1
SCHEMBL23280138 0.82 IDH1 (0.51) IDH1ROCK2ROCK1GPR84KDM4E
SCHEMBL19360603 0.81 MRGPRX4 (0.49) IDH1F2KDM4EALDH1A1LMNA
SCHEMBL19360302 0.79 KDM4E (0.43) F2KDM4EALDH1A1LMNAHTT
SCHEMBL30076020 0.79 KDM4E (0.43) F2KDM4EALDH1A1LMNAHTT
SCHEMBL978722 0.78 F2 (0.62) F2GPR84KDM4ELMNAKMT2A
SCHEMBL19360318 0.77 F2 (0.46) F2GPR84KDM4EALDH1A1LMNA
SCHEMBL19360546 0.76 MRGPRX4 (0.46) F2KDM4EALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531679-B Aromatic amide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed
CN-107531679-A Aromatic amides analog derivative, its preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-01-02 CN disclosed
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed