SCHEMBL19360696

SCHEMBL19360696

C=CC(=O)Nc1cccc(Nc2nc(Nc3ccccc3C)ncc2C)c1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BTK Q06187 6/20 0.82
EGFR P00533 16/20 0.77
ITK Q08881 5/20 0.77
MAPK3 P27361 1/20 0.61
JAK3 P52333 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9925020 0.92 BTK (0.79) BTKEGFRITKJAK3
SCHEMBL12519715 0.91 BTK (0.77) BTKEGFRITK
SCHEMBL2230183 0.90 BTK (1.00) BTKEGFRITKJAK3
SCHEMBL2352426 0.90 BTK (1.00) BTKEGFRITKJAK3
SCHEMBL9923759 0.89 EGFR (0.81) BTKEGFRITK
SCHEMBL13606336 0.87 EGFR (1.00) BTKEGFRITKJAK3
SCHEMBL2350876 0.87 EGFR (1.00) BTKEGFRITKJAK3
SCHEMBL2348879 0.87 EGFR (0.83) BTKEGFRITKMAPK3JAK3
SCHEMBL12518710 0.86 BTK (0.84) BTKEGFRITKJAK3
SCHEMBL28080977 0.86 BTK (0.88) BTKEGFRITKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9765038-B2 Heteroaryl compounds and uses thereof CELGENE CAR LLC (BM) 2017-09-19 US disclosed