SCHEMBL1936381

SCHEMBL1936381

CNC(=O)c1c(-c2ccc(F)cc2)oc2ncc(-c3cc(C(=O)N(c4ccccn4)C4CC4)ccc3C)cc12

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.53
CYP3A4 P08684 5/20 0.53
KCNH2 Q12809 3/20 0.53
NR1I2 O75469 1/20 0.53
ALDH1A1 P00352 3/20 0.45
TRPM8 Q7Z2W7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936895 0.93 CYP2C8 (0.54) CYP2C8CYP3A4KCNH2NR1I2
SCHEMBL2437777 0.92 ALDH1A1 (0.45) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL1935138 0.92 ALDH1A1 (0.47) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL2434818 0.91 ALDH1A1 (0.45) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL1918435 0.90 CYP2C8 (0.65) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL1936239 0.86 CYP2C8 (0.54) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL2433685 0.84 ALDH1A1 (0.45) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL1937242 0.83 ALDH1A1 (0.47) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL1919264 0.83 CYP2C8 (0.55) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1
SCHEMBL1918592 0.83 CYP2C8 (0.56) CYP2C8CYP3A4KCNH2NR1I2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545050-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112186-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed
EP-2331502-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2011-06-15 EP disclosed
WO-2010030538-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed