SCHEMBL19366286

SCHEMBL19366286

COc1cc2c(cc1C#N)CCC(C)[C@@H]2C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.48
AR P10275 4/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MAOA P21397 3/20 0.41
TSHR P16473 1/20 0.41
RAD52 P43351 1/20 0.38
DRD2 P14416 2/20 0.37
DRD1 P21728 2/20 0.37
KDM4E B2RXH2 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
BRD4 O60885 2/20 0.37
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17538345 1.00 HTR2A (0.48) HTR2AARCA1CA2MAOA
SCHEMBL6280381 0.77 HTR2C (0.52) HTR2ACA1CA2MAOATSHR
SCHEMBL16158423 0.77 MAOA (0.57) MAOATSHRDRD2DRD1ALDH1A1
SCHEMBL17538360 0.77 MAOA (0.44) CA1CA2MAOATSHRBRD4
SCHEMBL29741291 0.75 HTR2A (0.50) HTR2AARDRD2KDM4EUSP2
SCHEMBL16233593 0.74 HTR2A (0.48) HTR2AARKDM4EUSP2ALDH1A1
SCHEMBL25555806 0.74 HTR2A (0.51) HTR2AARKDM4EUSP2ALDH1A1
SCHEMBL19366293 0.73 HTR2A (0.45) HTR2AARCA1CA2DRD2
SCHEMBL19067966 0.73 HTR2A (0.45) HTR2AARCA1CA2DRD2
SCHEMBL15413032 0.73 MAOA (0.33) HTR2ACA1CA2MAOATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170266181-A1 NONSTEROIDAL AND STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-09-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170266181-A1 NONSTEROIDAL AND STEROIDAL COMPOUNDS WITH POTENT ANDROGEN RECEPTOR DOWN-REGULATION AND ANTI PROSTATE CANCER ACTIVITY AR, NR5A1, BRCA1 HTR2A 2253/4885AR 1/4885CA1 4054/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.