SCHEMBL19366609

SCHEMBL19366609

Cc1ccc(Nc2c(C(=O)NOC(CO)CO)cc3snnc3c2F)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 19/20 0.49
MAP2K2 P36507 5/20 0.40
ABCB11 O95342 1/20 0.40
NQO2 P16083 1/20 0.40
BRAF P15056 1/20 0.38
MAPK1 P28482 1/20 0.38
MAP2K5 Q13163 1/20 0.38
CSF1R P07333 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15131443 0.89 MAP2K1 (0.62) MAP2K1MAP2K2BRAFMAPK1MAP2K5
SCHEMBL15131347 0.89 MAP2K1 (0.49) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL19366605 0.87 MAP2K1 (0.54) MAP2K1MAP2K2ABCB11NQO2BRAF
SCHEMBL19367194 0.86 MAP2K1 (0.49) MAP2K1MAP2K2ABCB11NQO2BRAF
SCHEMBL19366603 0.86 MAP2K1 (0.53) MAP2K1MAP2K2ABCB11NQO2CYP3A4
SCHEMBL15131419 0.82 MAP2K1 (0.50) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL19367210 0.82 MEN1 (0.54) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL19367409 0.82 CSF1R (0.42) MAP2K1MAP2K2BRAFMAPK1CSF1R
SCHEMBL19367411 0.82 MAP2K1 (0.43) MAP2K1MAP2K2MAPK1CSF1R
SCHEMBL19366620 0.81 MAP2K1 (0.43) MAP2K1MAP2K2ABCB11NQO2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9937158-B2 Benzoheterocyclic compounds and use thereof SHANGHAI KECHOW PHARMA, INC. (CN) 2018-04-10 US disclosed
EP-2804855-B1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF SHANGHAI KECHOW PHARMA INC (CN) 2017-09-20 EP disclosed