SCHEMBL19367409

SCHEMBL19367409

COC(=O)c1cc2snnc2c(F)c1Nc1ccc(C)cc1F

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.42
MAPT P10636 1/20 0.39
MAP2K1 Q02750 7/20 0.36
MAP2K2 P36507 3/20 0.36
CYP46A1 Q9Y6A2 1/20 0.36
SCN5A Q14524 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
GFER P55789 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.35
RAF1 P04049 1/20 0.35
BRAF P15056 1/20 0.35
KCNH2 Q12809 4/20 0.35
MAPK1 P28482 1/20 0.35
SYK P43405 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19367411 0.89 MAP2K1 (0.43) CSF1RMAPTMAP2K1MAP2K2MEN1
SCHEMBL15130253 0.88 MAP2K1 (0.48) MAP2K1MAP2K2BRAFMAPK1
SCHEMBL15130159 0.87 NPC1 (0.43) CSF1RMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL19366595 0.83 CSF1R (0.44) CSF1RMAP2K1MAP2K2CYP46A1MEN1
SCHEMBL19366603 0.83 MAP2K1 (0.53) MAP2K1MAP2K2
SCHEMBL19366609 0.82 MAP2K1 (0.49) CSF1RMAP2K1MAP2K2BRAFMAPK1
SCHEMBL15130261 0.81 USP2 (0.41) CSF1RMAPTSMN1; SMN2ALDH1A1
SCHEMBL15130290 0.81 MAP2K1 (0.45) CSF1RMAPTMAP2K1MAP2K2ALDH1A1
SCHEMBL19367210 0.80 MEN1 (0.54) MAP2K1MAP2K2MEN1KMT2ARAF1
SCHEMBL19366605 0.80 MAP2K1 (0.54) MAP2K1MAP2K2BRAFMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9937158-B2 Benzoheterocyclic compounds and use thereof SHANGHAI KECHOW PHARMA, INC. (CN) 2018-04-10 US disclosed
EP-2804855-B1 BENZOHETEROCYCLIC COMPOUNDS AND USE THEREOF SHANGHAI KECHOW PHARMA INC (CN) 2017-09-20 EP disclosed