SCHEMBL1936737

SCHEMBL1936737

COC(=O)Oc1cc(Oc2cc(C(=O)Nc3cc(C(C)(C)C)cc(NS(C)(=O)=O)c3OC)ccc2C)ccn1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRAF P15056 14/20 0.52
GSK3A P49840 4/20 0.50
MAPK14 Q16539 3/20 0.46
LCK P06239 2/20 0.46
SRC P12931 2/20 0.46
SYK P43405 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1936086 0.92 GSK3A (0.49) BRAFGSK3AMAPK14LCKSRC
SCHEMBL1936661 0.89 BRAF (0.57) BRAF
SCHEMBL1936147 0.88 BRAF (0.54) BRAFGSK3AMAPK14LCKSRC
SCHEMBL2671306 0.88 BRAF (0.54) BRAFGSK3AMAPK14LCKSRC
SCHEMBL15062881 0.87 GSK3A (0.56) BRAFGSK3AMAPK14LCKSRC
SCHEMBL1934863 0.87 BRAF (0.55) BRAFGSK3AMAPK14
SCHEMBL1936181 0.87 BRAF (0.53) BRAFMAPK14
SCHEMBL1936373 0.87 BRAF (0.52) BRAFGSK3AMAPK14LCKSRC
SCHEMBL1936240 0.85 BRAF (0.51) BRAFGSK3AMAPK14LCKSRC
SCHEMBL1934475 0.83 BRAF (0.56) BRAFGSK3AMAPK14SRCSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2331506-B1 NOVEL BENZAMIDES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INT (DE) 2013-07-03 EP disclosed
EP-2331506-A1 NOVEL BENZAMIDES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS Boehringer Ingelheim International GmbH (DE) 2011-06-15 EP disclosed
WO-2010026095-A1 NOVEL BENZAMIDES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-03-11 WO disclosed