SCHEMBL1937087

SCHEMBL1937087

Cc1ccc(C(=O)NC2(c3ccccc3)CC2)cc1N(C)C(=O)c1c(-c2ccc(F)cc2)nn2c(F)cccc12

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.44
CYP3A4 P08684 5/20 0.44
DGAT2 Q96PD7 6/20 0.37
TACR1 P25103 1/20 0.36
KCNH2 Q12809 3/20 0.36
NR1I2 O75469 1/20 0.36
TTK P33981 1/20 0.35
PTGER4 P35408 2/20 0.34
TACR3 P29371 1/20 0.34
MAPK14 Q16539 1/20 0.33
IDO1 P14902 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464955 0.77 CYP2C8 (0.60) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL2463689 0.77 CYP2C8 (0.46) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL1936906 0.74 NPC1 (0.42) CYP2C8CYP3A4IDO1
SCHEMBL2464836 0.74 CYP2C8 (0.60) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL9911902 0.72 CYP2C8 (0.62) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL13241638 0.71 CYP2C8 (0.59) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL13459293 0.71 CYP2C8 (0.53) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL1935064 0.71 CYP2C8 (0.46) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL666705 0.71 CYP2C8 (0.46) CYP2C8CYP3A4DGAT2KCNH2NR1I2
SCHEMBL1937117 0.70 CYP2C8 (0.57) CYP2C8CYP3A4DGAT2KCNH2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2331502-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2011-06-15 EP disclosed
WO-2010030538-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed