SCHEMBL19387993

SCHEMBL19387993

CC(C)(C)NC(=O)Cc1cncnc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
HPGD P15428 2/20 0.41
CYP2C9 P11712 1/20 0.41
ANO1 Q5XXA6 4/20 0.41
KDM4E B2RXH2 2/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 1/20 0.39
PDE4B Q07343 1/20 0.38
POLB P06746 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2757955 0.80 CYP1A2 (0.69) CA1CA2CYP1A2CYP3A4CYP2C9
SCHEMBL1484349 0.79 CYP1A2 (0.41) CYP1A2CYP3A4CYP2C9RAB9APOLB
SCHEMBL19133623 0.78 CA1 (0.59) CA1CA2HPGDANO1KDM4E
SCHEMBL19387994 0.78 RAB9A (0.58) CA1CA2HPGDANO1KDM4E
SCHEMBL25434734 0.76 HDAC6 (0.52) CYP1A2CYP3A4CYP2C9KDM4E
SCHEMBL16891683 0.76 GAA (0.39) CYP1A2CYP3A4HPGDCYP2C9L3MBTL1
SCHEMBL16886387 0.75 HCAR2 (0.37) CYP1A2CYP3A4CYP2C9RAB9AMAPT
SCHEMBL25404860 0.74 HTT (0.41) CYP1A2CYP3A4CYP2C9KDM4ELMNA
SCHEMBL19387992 0.74 CA1 (0.48) CA1CA2CYP1A2CYP3A4HPGD
SCHEMBL8240261 0.73 HPGD (0.71) CA1CA2HPGDANO1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9771320-B2 Carbocyclic sulfone RORγ modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2017-09-26 US disclosed