SCHEMBL19412840

SCHEMBL19412840

C[C@H](c1ccccc1)C1CCN([C@@H](C)c2ccccc2)C1=O

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
MCOLN3 Q8TDD5 1/20 0.50
KMT2A Q03164 1/20 0.49
HPGD P15428 1/20 0.48
CYP2D6 P10635 1/20 0.46
MAPK1 P28482 1/20 0.45
HSD11B1 P28845 2/20 0.45
GAA P10253 1/20 0.43
PKM P14618 1/20 0.41
MC4R P32245 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14177729 1.00 ALDH1A1 (0.50) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL14177730 1.00 ALDH1A1 (0.50) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL14195929 1.00 ALDH1A1 (0.50) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL14177728 1.00 ALDH1A1 (0.50) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL19412900 1.00 ALDH1A1 (0.50) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL5629867 0.86 KMT2A (0.48) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL5629865 0.86 KMT2A (0.48) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL14177732 0.86 KMT2A (0.43) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL14177733 0.86 KMT2A (0.43) ALDH1A1MCOLN3KMT2AHPGDCYP2D6
SCHEMBL14196200 0.86 KMT2A (0.43) ALDH1A1MCOLN3KMT2AHPGDCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9776965-B2 Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors JANSSEN PHARMACEUTICA NV (BE) 2017-10-03 US disclosed